SCHEMBL28610367

SCHEMBL28610367

Cc1[nH]c(C)c(C(=O)O)c1C.O=C1Cc2ccc(-c3cccnc3)cc2N1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 12/20 0.56
CYP11B2 P19099 12/20 0.56
CYP1A2 P05177 3/20 0.56
TDP2 O95551 2/20 0.51
CYP2C9 P11712 2/20 0.47
TBXAS1 P24557 1/20 0.47
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
CRBN Q96SW2 2/20 0.46
CYP19A1 P11511 3/20 0.43
FABP7 O15540 1/20 0.41
FABP3 P05413 1/20 0.41
FABP5 Q01469 1/20 0.41
CYP3A4 P08684 2/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
CYP2C19 P33261 1/20 0.41
DHODH Q02127 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28606058 0.90 CRBN (0.53) CYP11B1CYP11B2CYP1A2TDP2CRBN
SCHEMBL29899622 0.82 CYP11B1 (0.79) CYP11B1CYP11B2CYP1A2TDP2CYP2C9
SCHEMBL3659028 0.82 CYP11B1 (0.79) CYP11B1CYP11B2CYP1A2TDP2CYP2C9
SCHEMBL28607397 0.82 CRBN (0.48) TDP2CRBNFABP7FABP3FABP5
SCHEMBL28918955 0.82 FABP7 (0.52) TDP2CRBNFABP7FABP3FABP5
SCHEMBL28595556 0.81 GRIA1 (0.53) CYP11B1CYP11B2CYP1A2TDP2PDE3B
SCHEMBL29016191 0.74 CRBN (0.54) TDP2CRBNFABP7FABP3FABP5
SCHEMBL29849827 0.73 CYP11B1 (1.00) CYP11B1CYP11B2CYP1A2TDP2CYP2C9
SCHEMBL748904 0.73 CYP11B1 (1.00) CYP11B1CYP11B2CYP1A2TDP2CYP2C9
SCHEMBL29899595 0.73 CYP11B1 (1.00) CYP11B1CYP11B2CYP1A2TDP2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113181362-A Agent for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2021-07-30 CN disclosed