SCHEMBL28611549

SCHEMBL28611549

Cc1ccnc(C(C)C)c1NC(=O)C(C#N)C(=O)c1cc(F)c(Cl)nc1Cl

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
MAP4K1 Q92918 1/20 0.33
DHODH Q02127 4/20 0.32
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KRAS P01116 1/20 0.30
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30800345 1.00 KEAP1 (0.35) KEAP1NFE2L2MAP4K1DHODHLMNA
SCHEMBL23830113 0.90 MAP4K1 (0.33) MAP4K1KRAS
SCHEMBL28599872 0.81 DHODH (0.37) KEAP1NFE2L2DHODH
SCHEMBL29742278 0.79 GAA (0.39) KEAP1NFE2L2DHODHLMNASMN1; SMN2
SCHEMBL20560749 0.79 GAA (0.39) KEAP1NFE2L2DHODHLMNASMN1; SMN2
SCHEMBL29742271 0.79 GAA (0.39) KEAP1NFE2L2DHODHLMNASMN1; SMN2
SCHEMBL28599875 0.77 DHODH (0.35) KEAP1NFE2L2DHODH
SCHEMBL24502503 0.73 KEAP1 (0.36) KEAP1NFE2L2DHODHKRAS
SCHEMBL25415392 0.73 KEAP1 (0.43) KEAP1NFE2L2DHODHLMNASMN1; SMN2
SCHEMBL29572702 0.73 KEAP1 (0.43) KEAP1NFE2L2DHODHLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113286794-B KRAS mutein inhibitors 北京加科思新药研发有限公司 2024-03-12 CN disclosed
CN-113286794-A KRAS mutein inhibitors 北京加科思新药研发有限公司 2021-08-20 CN disclosed