SCHEMBL28599872

SCHEMBL28599872

CCOC(=O)C(C(=O)Nc1c(C)ccnc1C(C)C)C(=O)c1cc(F)c(Cl)nc1Cl

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 10/20 0.37
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
NLRP3 Q96P20 1/20 0.32
PIK3C3 Q8NEB9 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
PKM P14618 1/20 0.31
KMT2A Q03164 1/20 0.31
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28599875 0.90 DHODH (0.35) DHODHKEAP1NFE2L2KMT2A
SCHEMBL28611549 0.81 KEAP1 (0.35) DHODHKEAP1NFE2L2
SCHEMBL30800345 0.81 KEAP1 (0.35) DHODHKEAP1NFE2L2
SCHEMBL20560749 0.78 GAA (0.39) DHODHKEAP1NFE2L2NPC1RAB9A
SCHEMBL29742278 0.78 GAA (0.39) DHODHKEAP1NFE2L2NPC1RAB9A
SCHEMBL29742271 0.78 GAA (0.39) DHODHKEAP1NFE2L2NPC1RAB9A
SCHEMBL9686323 0.78 KEAP1 (0.51) KEAP1NFE2L2NPC1MAPTRAB9A
SCHEMBL25414127 0.76 DHODH (0.34) DHODH
SCHEMBL31020499 0.76 DHODH (0.33) DHODHNLRP3PKM
SCHEMBL29962647 0.76 DHODH (0.34) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112920183-A Compounds as KRAS-G12C inhibitors and uses thereof 南京圣和药业股份有限公司 2021-06-08 CN disclosed