SCHEMBL28613325

SCHEMBL28613325

CC(C)(C)OC(=O)N[C@@H](CC#CBr)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.48
CTSK P43235 10/20 0.48
CTSL P07711 2/20 0.46
CTSB P07858 2/20 0.46
PPARA Q07869 5/20 0.43
PPARG P37231 4/20 0.43
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
ACE P12821 1/20 0.42
PPARD Q03181 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28613327 1.00 CTSS (0.48) CTSSCTSKCTSLCTSBPPARA
SCHEMBL28961693 0.86 CTSK (0.44) CTSSCTSKCTSLCTSB
SCHEMBL22109891 0.86 CTSK (0.44) CTSSCTSKCTSLCTSB
SCHEMBL1429918 0.86 CTSK (0.61) CTSSCTSKCTSLCTSBPPARA
SCHEMBL2399357 0.86 CTSK (0.61) CTSSCTSKCTSLCTSBPPARA
SCHEMBL1429799 0.86 CTSK (0.61) CTSSCTSKCTSLCTSBPPARA
SCHEMBL17533115 0.82 CTSS (0.46) CTSSCTSKCTSLCTSBPPARA
SCHEMBL1952503 0.81 CTSS (0.61) CTSSCTSKCTSLCTSB
SCHEMBL999757 0.81 CTSS (0.61) CTSSCTSKCTSLCTSB
SCHEMBL17708331 0.81 CTSS (0.61) CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113195473-B Tricyclic compound as STING agonist and preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113195473-A Tricyclic compound as STING agonist and preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-30 CN disclosed