SCHEMBL28614908

SCHEMBL28614908

CC(C)(C)NC(=O)O[C@H]1CC(=O)NC1=O

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.34
CRBN Q96SW2 7/20 0.33
DDB1 Q16531 6/20 0.33
TSHR P16473 2/20 0.33
MAPK1 P28482 1/20 0.33
MAP3K14 Q99558 1/20 0.32
GBA1 P04062 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28864213 1.00 GAA (0.34) GAACRBNDDB1TSHRMAPK1
SCHEMBL4773108 0.84 DDB1 (0.46) CRBNDDB1
SCHEMBL1773976 0.77 CRBN (0.40) GAACRBNDDB1MAPK1MAP3K14
SCHEMBL756451 0.76 CRBN (0.38) GAACRBNDDB1TSHRMAP3K14
SCHEMBL8576306 0.76 EPHX2 (0.42) GAA
SCHEMBL10633587 0.76 EPHX2 (0.42) GAA
SCHEMBL57232 0.75 MAP3K14 (0.39) GAACRBNDDB1TSHRMAP3K14
SCHEMBL28585016 0.75 LMNA (0.31) GAA
SCHEMBL3836555 0.75 EPHX2 (0.40) GAACRBNDDB1TSHR
SCHEMBL27675961 0.75 IDO1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153644-B Small molecules against CEREBLON to enhance effector T cell function H·李·莫菲特癌症中心研究有限公司 2022-10-21 CN disclosed
CN-112512589-A Dimeric immunomodulatory compounds against CEREBLON-based mechanisms H·李·莫菲特癌症中心研究有限公司 2021-03-16 CN disclosed
CN-109153644-A SMALL MOLECULES AGAINST CEREBLON TO ENHANCE EFFECTOR T CELL FUNCTION H·李·莫菲特癌症中心研究有限公司 2019-01-04 CN disclosed