SCHEMBL28616101

SCHEMBL28616101

Fc1ccc(N2CCc3ccccc3C2C#Cc2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
GAA P10253 1/20 0.39
PRCP P42785 2/20 0.38
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
DRD2 P14416 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
DRD1 P21728 1/20 0.37
DRD4 P21917 1/20 0.37
ADRA1D P25100 1/20 0.37
HTR2A P28223 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
DRD3 P35462 1/20 0.37
HTR2B P41595 1/20 0.37
KCNH2 Q12809 12/20 0.36
SLC6A4 P31645 1/20 0.35
CCR3 P51677 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30168542 1.00 ESR1 (0.42) ESR1ESR2GAAPRCPHTR1A
SCHEMBL30168543 0.90 ESR1 (0.39) ESR1ESR2GAAPRCP
SCHEMBL28615700 0.90 ESR1 (0.39) ESR1ESR2GAAPRCP
SCHEMBL30168540 0.88 PRCP (0.38) ESR1ESR2PRCP
SCHEMBL28632888 0.88 PRCP (0.38) ESR1ESR2PRCP
SCHEMBL30168541 0.87 PRCP (0.38) ESR1ESR2GAAPRCP
SCHEMBL28619047 0.87 PRCP (0.38) ESR1ESR2GAAPRCP
SCHEMBL28632884 0.86 TRPM8 (0.39) PRCP
SCHEMBL30168545 0.86 TRPM8 (0.39) PRCP
SCHEMBL28625714 0.82 ESR1 (0.44) ESR1ESR2GAAPRCPHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307769-B 1-alkynyl tetrahydroisoquinoline compound and preparation method thereof 长江师范学院 2023-03-03 CN disclosed
CN-113307769-A 1-alkynyl tetrahydroisoquinoline compound and preparation method thereof 长江师范学院 2021-08-27 CN disclosed