SCHEMBL28632884

SCHEMBL28632884

FC(F)(F)c1ccc(N2CCc3ccccc3C2C#Cc2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 14/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
KDM4E B2RXH2 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
OPRD1 P41143 1/20 0.37
PRCP P42785 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30168545 1.00 TRPM8 (0.39) TRPM8HDAC3HDAC1HDAC8NCOR2
SCHEMBL28615700 0.87 ESR1 (0.39) PRCP
SCHEMBL30168543 0.87 ESR1 (0.39) PRCP
SCHEMBL28616101 0.86 ESR1 (0.42) PRCP
SCHEMBL30168542 0.86 ESR1 (0.42) PRCP
SCHEMBL30101766 0.85 TRPM8 (0.43) TRPM8HDAC3HDAC1HDAC8NCOR2
SCHEMBL28632888 0.85 PRCP (0.38) HDAC3HDAC1HDAC8NCOR2PRCP
SCHEMBL28630559 0.85 TRPM8 (0.43) TRPM8HDAC3HDAC1HDAC8NCOR2
SCHEMBL30168540 0.85 PRCP (0.38) HDAC3HDAC1HDAC8NCOR2PRCP
SCHEMBL30168541 0.84 PRCP (0.38) KDM4EPRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307769-B 1-alkynyl tetrahydroisoquinoline compound and preparation method thereof 长江师范学院 2023-03-03 CN disclosed
CN-113307769-A 1-alkynyl tetrahydroisoquinoline compound and preparation method thereof 长江师范学院 2021-08-27 CN disclosed