SCHEMBL28616232

SCHEMBL28616232

C=CC(=O)Nc1ccc(C(=O)NCc2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.59
HDAC2 Q92769 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
TGM2 P21980 3/20 0.58
HPGD P15428 1/20 0.56
LMNA P02545 1/20 0.55
RAB9A P51151 1/20 0.55
TP53 P04637 1/20 0.54
MAPT P10636 1/20 0.54
HDAC1 Q13547 2/20 0.54
ROCK2 O75116 1/20 0.52
RPS6KA5 O75582 1/20 0.52
MAP4K4 O95819 1/20 0.52
PRKCG P05129 1/20 0.52
PRKACA P17612 1/20 0.52
RPS6KB1 P23443 1/20 0.52
MAPK1 P28482 1/20 0.52
AKT1 P31749 1/20 0.52
GSK3A P49840 1/20 0.52
GSK3B P49841 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11775423 0.85 TGM2 (0.71) TGM2HPGDLMNARAB9ATP53
SCHEMBL17744942 0.83 HDAC6 (0.68) HDAC6HDAC2HDAC8HPGDLMNA
SCHEMBL29635001 0.82 TGM2 (0.66) TGM2LMNACA2
SCHEMBL11900090 0.81 HDAC6 (0.85) HDAC6HDAC2HDAC8HPGDLMNA
SCHEMBL18601428 0.79 KMT2A (0.68) HDAC6HDAC2HDAC8HPGDLMNA
SCHEMBL28648926 0.79 HDAC6 (0.70) HDAC6HDAC2HDAC8HPGDLMNA
SCHEMBL29157753 0.79 TGM2 (0.70) TGM2LMNACA2POLB
Hydrochloric Acid SCHEMBL27676561 0.78 NSD2 (0.50) TGM2HPGDLMNAKDM4E
SCHEMBL40744 0.78 TGM2 (0.68) TGM2HPGDLMNATSHR
SCHEMBL17327878 0.78 TGM2 (0.63) TGM2LMNARAB9AKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109438279-B Small molecule compound for overcoming EGFR drug-resistant mutation and preparation method and application thereof 四川大学 2021-08-31 CN disclosed