SCHEMBL28616617

SCHEMBL28616617

Nc1nc(-c2ccccc2)c(CNS(=O)(=O)c2ccc(F)cc2)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
ALDH1A1 P00352 4/20 0.49
MAPT P10636 2/20 0.49
KIT P10721 1/20 0.48
CYP19A1 P11511 1/20 0.45
KMT2A Q03164 2/20 0.44
TAAR1 Q96RJ0 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
TP53 P04637 1/20 0.44
THRB P10828 1/20 0.44
NPSR1 Q6W5P4 2/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
PTGS2 P35354 1/20 0.42
PTGDR2 Q9Y5Y4 2/20 0.42
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28633647 0.88 MAPT (0.55) ALDH1A1MAPTKITKMT2ACA1
SCHEMBL28618016 0.88 ALDH1A1 (0.55) CYP1A2ALDH1A1MAPTCYP19A1KMT2A
SCHEMBL28615807 0.88 ALDH1A1 (0.53) CYP1A2ALDH1A1MAPTCYP19A1KMT2A
SCHEMBL28631505 0.85 MAPT (0.55) CYP1A2ALDH1A1MAPTCYP19A1KMT2A
SCHEMBL28621324 0.85 MEN1 (0.57) CYP1A2ALDH1A1MAPTCYP19A1KMT2A
SCHEMBL28627987 0.81 ALDH1A1 (0.56) CYP1A2ALDH1A1MAPTCYP19A1KMT2A
SCHEMBL28922648 0.78 THRB (0.55) CYP1A2ALDH1A1MAPTCYP19A1KMT2A
SCHEMBL28616619 0.77 SMN1; SMN2 (0.50) CYP1A2ALDH1A1MAPTCYP19A1KMT2A
SCHEMBL28619745 0.77 HTT (0.52) ALDH1A1MAPTKMT2ANPSR1MEN1
SCHEMBL28616278 0.77 ALDH1A1 (0.44) CYP1A2ALDH1A1MAPTCYP19A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113214183-A 5- (aminomethyl) -4-arylthiophene-2-amine derivative and preparation method thereof 上海应用技术大学 2021-08-06 CN disclosed