SCHEMBL28617952

SCHEMBL28617952

O=C(Nc1cccc(Br)c1F)C1CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.50
HPGD P15428 2/20 0.49
KMT2A Q03164 2/20 0.48
PLAU P00749 1/20 0.47
NPC1 O15118 1/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
CASP3 P42574 1/20 0.46
CETP P11597 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
ALOX15 P16050 1/20 0.44
ALOX12 P18054 1/20 0.44
HTT P42858 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31381754 1.00 TP53 (0.50) TP53HPGDKMT2APLAUNPC1
SCHEMBL28669892 0.83 NPC1 (0.63) TP53HPGDKMT2ANPC1GAA
SCHEMBL123452 0.81 LMNA (0.51) TP53HPGDPLAUNPC1GAA
SCHEMBL3415512 0.78 KMT2A (0.49) TP53KMT2ANPC1SMN1; SMN2ALDH1A1
SCHEMBL27839469 0.77 PLAU (0.47) HPGDKMT2APLAUNPC1GAA
SCHEMBL5699255 0.77 GAA (0.44) HPGDPLAUNPC1GAAPKM
SCHEMBL20560218 0.76 HTT (0.46) TP53HPGDKMT2ANPC1GAA
SCHEMBL146375 0.76 RXFP1 (0.50) HPGDKMT2ANPC1GAAHDAC1
SCHEMBL4744831 0.76 SMN1; SMN2 (0.67) KMT2ANPC1GAAPKMCETP
SCHEMBL18554486 0.76 CTSC (0.42) TP53KMT2ASMN1; SMN2MEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113015526-A Spirocyclic 2, 3-dihydro-7-azaindole compounds and uses thereof 豪夫迈·罗氏有限公司 2021-06-22 CN disclosed