SCHEMBL28619948

SCHEMBL28619948

Cn1c(=O)c2c(nc(OCCCOc3ccccc3)n2C)n(C)c1=O

nearest known ligand 0.93

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOA P21397 13/20 0.93
MAOB P27338 13/20 0.93
KMT2A Q03164 1/20 0.73
PKM P14618 2/20 0.70
HTT P42858 2/20 0.70
SMN1; SMN2 Q16637 2/20 0.64
HSD17B10 Q99714 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28886844 0.95 MAOA (0.84) MAOAMAOBKMT2APKMHTT
SCHEMBL28623824 0.90 MAOA (0.75) MAOAMAOBKMT2APKMHTT
SCHEMBL28629790 0.89 MAOA (0.74) MAOAMAOBKMT2APKMHTT
SCHEMBL28615788 0.85 MAOB (0.69) MAOAMAOBKMT2APKMHTT
SCHEMBL28625191 0.85 MAOA (0.69) MAOAMAOBKMT2APKMHTT
SCHEMBL28634494 0.84 TSHR (0.74) MAOAMAOBKMT2APKMHTT
SCHEMBL28921780 0.82 MAOA (0.65) MAOAMAOBKMT2APKMSMN1; SMN2
SCHEMBL28622147 0.81 MAOA (0.70) MAOAMAOBKMT2APKMSMN1; SMN2
SCHEMBL29987280 0.80 MAOA (0.61) MAOAMAOBKMT2APKMSMN1; SMN2
SCHEMBL19994563 0.79 MAOB (1.00) MAOAMAOBPKMHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354646-B 8-aryloxy alkoxy substituted xanthine derivative and preparation method and application thereof 南开大学 2022-11-15 CN claimed
CN-113354646-A 8-aryloxy alkoxy substituted xanthine derivative and preparation method and application thereof 南开大学 2021-09-07 CN claimed
CN-113354646-B 8-aryloxy alkoxy substituted xanthine derivative and preparation method and application thereof 南开大学 2022-11-15 CN disclosed
CN-113354646-A 8-aryloxy alkoxy substituted xanthine derivative and preparation method and application thereof 南开大学 2021-09-07 CN disclosed