SCHEMBL2862215

SCHEMBL2862215

FC(F)(F)c1ccc(CCNc2ncnc3c2CNCC3)cn1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 10/20 0.45
P2RX2 Q9UBL9 7/20 0.45
GRIN2B Q13224 2/20 0.38
MCHR1 Q99705 4/20 0.38
DAO P14920 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2866604 0.89 P2RX3 (0.55) P2RX3P2RX2MCHR1CNR1CNR2
SCHEMBL2868273 0.81 HTR2C (0.48)
SCHEMBL4339725 0.80 TTBK1 (0.51) CNR1CNR2
SCHEMBL2847817 0.79 APP (0.41)
SCHEMBL2867255 0.75 P2RX3 (0.55) P2RX3P2RX2
SCHEMBL4759238 0.74 P2RX3 (0.58) P2RX3P2RX2
SCHEMBL2857789 0.74 P2RX3 (0.36) P2RX3P2RX2GRIN2BMCHR1
SCHEMBL2862214 0.74 P2RX3 (0.58) P2RX3P2RX2
SCHEMBL4340134 0.73 P2RX3 (0.65) P2RX3P2RX2
SCHEMBL4341209 0.73 P2RX3 (0.66) P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139334-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2010-01-06 EP disclosed
WO-2008130481-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2008-10-30 WO disclosed