SCHEMBL28623788

SCHEMBL28623788

CC(C(O)C#N)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.45
KMT2A Q03164 3/20 0.45
GAA P10253 1/20 0.45
NPBWR1 P48145 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MCHR1 Q99705 1/20 0.45
ALDH1A1 P00352 4/20 0.44
SIGMAR1 Q99720 1/20 0.41
MEN1 O00255 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
SLC6A2 P23975 2/20 0.40
HTR2A P28223 2/20 0.40
ADRA1A P35348 2/20 0.40
SLC6A3 Q01959 2/20 0.40
KCNH2 Q12809 2/20 0.40
SLC6A4 P31645 1/20 0.40
OPRK1 P41145 1/20 0.40
MMP1 P03956 4/20 0.39
MMP3 P08254 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17275467 1.00 TSHR (0.45) TSHRKMT2AGAANPBWR1NPSR1
SCHEMBL531663 0.82 MEN1 (0.51) KMT2AALDH1A1MEN1MMP1MMP3
SCHEMBL4369852 0.80 TSHR (0.43) TSHRKMT2AGAANPBWR1NPSR1
SCHEMBL26989268 0.80 TSHR (0.46) TSHRKMT2AGAANPBWR1NPSR1
SCHEMBL26988083 0.80 TSHR (0.46) TSHRKMT2AGAANPBWR1NPSR1
SCHEMBL26988540 0.80 TSHR (0.46) TSHRKMT2AGAANPBWR1NPSR1
SCHEMBL428101 0.80 TSHR (0.46) TSHRKMT2AGAANPBWR1NPSR1
SCHEMBL26987985 0.80 TSHR (0.46) TSHRKMT2AGAANPBWR1NPSR1
SCHEMBL2565075 0.78 ALDH1A1 (0.50) TSHRKMT2AGAANPBWR1NPSR1
SCHEMBL5872219 0.78 TSHR (0.44) TSHRKMT2AGAANPBWR1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106661084-B Macrocyclic broad spectrum antibiotics 阿奇克斯制药公司 2021-08-31 CN disclosed
CN-106661084-A Macrocyclic broad spectrum antibiotics 阿奇克斯制药公司 2017-05-10 CN disclosed