SCHEMBL28624352

SCHEMBL28624352

O=C(O)c1cc2nc[nH]c(=O)c2cc1-c1cccc(F)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOD1 Q9Y239 4/20 0.56
PARP1 P09874 3/20 0.50
NOD2 Q9HC29 1/20 0.48
TEK Q02763 3/20 0.46
MAPKAPK2 P49137 1/20 0.44
ACVR1 Q04771 2/20 0.44
KDR P35968 1/20 0.43
EPHB4 P54760 1/20 0.43
GPR35 Q9HC97 2/20 0.43
KMO O15229 2/20 0.42
AXL P30530 1/20 0.42
DHODH Q02127 1/20 0.41
IP6K1 Q92551 1/20 0.41
IP6K3 Q96PC2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28622745 0.86 NOD1 (0.57) NOD1PARP1NOD2TEKACVR1
SCHEMBL6921163 0.77 TEK (0.59) PARP1TEKMAPKAPK2ACVR1KDR
SCHEMBL28128312 0.73 PARP1 (0.59) PARP1MAPKAPK2ACVR1
SCHEMBL4141791 0.71 IP6K1 (0.52) PARP1IP6K1IP6K3
SCHEMBL4141934 0.71 SLC2A1 (0.54) PARP1ACVR1IP6K1IP6K3
SCHEMBL4148739 0.71 PARP1 (0.51) PARP1ACVR1IP6K1IP6K3
SCHEMBL28619439 0.71 NOD1 (0.68) NOD1NOD2
SCHEMBL17797037 0.70 DCLRE1B (0.56) KDRGPR35KMODHODH
SCHEMBL17796982 0.70 DCLRE1B (0.53) KDRGPR35KMODHODH
SCHEMBL31585756 0.70 DCLRE1B (0.53) KDRGPR35KMODHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354590-A Quinazolinone compound for antagonizing NOD1/2 receptor signal pathway 宁波康柏睿格医药科技有限公司 2021-09-07 CN disclosed