SCHEMBL28625477

SCHEMBL28625477

Cc1cc(NC(=O)C(N)=O)ccc1C(=O)N1CCCC(=O)c2cc(Cl)ccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 14/20 0.51
AVPR1A P37288 2/20 0.51
ABCB11 O95342 1/20 0.51
ADRB2 P07550 1/20 0.51
HTR1A P08908 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
CHRM1 P11229 1/20 0.51
TBXA2R P21731 1/20 0.51
HTR2C P28335 1/20 0.51
HRH1 P35367 1/20 0.51
OPRM1 P35372 1/20 0.51
GLP1R P43220 1/20 0.51
TMEM97 Q5BJF2 1/20 0.51
FFAR4 Q5NUL3 1/20 0.51
GPR119 Q8TDV5 1/20 0.51
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28625478 0.90 AVPR2 (0.49) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL533754 0.85 AVPR2 (0.70) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL31344362 0.85 AVPR2 (0.70) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL30354671 0.85 AVPR2 (0.70) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL1291366 0.83 AVPR2 (0.71) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL29776619 0.83 AVPR2 (0.51) AVPR2AVPR1AABCB11ADRB2HTR1A
Hydrochloric Acid SCHEMBL30354670 0.83 AVPR2 (0.70) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL28617462 0.82 AVPR2 (0.75) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL24103986 0.81 AVPR2 (0.53) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL30354669 0.81 AVPR2 (0.53) AVPR2AVPR1AABCB11ADRB2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113277980-B Tolvaptan impurity and preparation method thereof 南京海纳医药科技股份有限公司 2022-09-02 CN disclosed
CN-113277980-A Tolvaptan impurity and preparation method thereof 南京海纳医药科技股份有限公司 2021-08-20 CN disclosed