SCHEMBL28626495

SCHEMBL28626495

CCN(CC)Cc1ccc(NC(=O)c2cc3cccc(O)c3oc2=O)cc1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 7/20 0.61
AR P10275 4/20 0.61
MAPT P10636 3/20 0.56
TP53 P04637 2/20 0.56
MAOA P21397 4/20 0.55
MAOB P27338 4/20 0.55
CBR1 P16152 3/20 0.53
AKR1B10 O60218 1/20 0.52
AKR1B1 P15121 1/20 0.52
MEN1 O00255 1/20 0.52
POLB P06746 1/20 0.52
KMT2A Q03164 1/20 0.52
PLEC Q15149 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
AKR1C1 Q04828 1/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28636450 0.91 POLB (0.53) AKR1C3ARMAPTTP53MAOA
SCHEMBL28626506 0.89 AKR1C3 (0.60) AKR1C3ARMAPTTP53MAOA
SCHEMBL28630607 0.88 MAPT (0.74) MAPTTP53MEN1POLBKMT2A
SCHEMBL28621873 0.81 HSD17B1 (0.48) AKR1C3ARMAPTTP53MAOA
SCHEMBL28621586 0.81 POLB (0.53) AKR1C3ARMAPTTP53MAOA
SCHEMBL28625763 0.80 MAPT (0.62) MAPTTP53MEN1POLBKMT2A
SCHEMBL28641067 0.77 MAPT (0.76) MAPTTP53MEN1POLBKMT2A
SCHEMBL28636610 0.76 AKR1C3 (0.52) AKR1C3ARMAPTTP53MAOA
SCHEMBL3880564 0.75 MAPT (0.77) MAPTTP53MEN1POLBKMT2A
SCHEMBL28865516 0.74 MAOA (0.68) AKR1C3MAPTMAOAMAOBAKR1B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108715589-B Coumarin derivative used as caspase-3 activator and application thereof 华侨大学 2021-04-20 CN disclosed