SCHEMBL28626849

SCHEMBL28626849

C[C@H](CCF)N(C)C(=O)c1cc2ccccc2c(-c2cnccc2Cl)n1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSPO P30536 7/20 0.63
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2C9 P11712 1/20 0.63
TSHR P16473 1/20 0.63
ALDH1A1 P00352 1/20 0.63
BLM P54132 1/20 0.63
PMP22 Q01453 1/20 0.63
NR1I3 Q14994 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28626851 1.00 TSPO (0.63) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8473060 0.81 TSPO (0.79) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8471215 0.78 TSPO (0.59) TSPOMEN1KMT2ACYP3A4CYP2C9
Pk-11195 SCHEMBL29354252 0.78 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
Pk-11195 SCHEMBL31060347 0.78 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL12790424 0.78 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL29357086 0.78 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL29477174 0.78 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL15118334 0.78 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9
(R)Pk-11195 SCHEMBL3126094 0.78 TSPO (1.00) TSPOMEN1KMT2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113387896-B 4- (2-chloro aryl) quinazoline-2-amide derivative and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2023-03-24 CN disclosed
CN-113387896-A 4- (2-chloro aryl) quinazoline-2-amide derivative and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2021-09-14 CN disclosed