SCHEMBL28628874

SCHEMBL28628874

CC(C)(C)OC(=O)Nc1ccc(C(N)=O)cc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.46
AAK1 Q2M2I8 7/20 0.46
CYP17A1 P05093 1/20 0.46
PRKCI P41743 1/20 0.43
MAPT P10636 4/20 0.43
GAA P10253 2/20 0.43
MAPK1 P28482 1/20 0.43
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HSD17B10 Q99714 1/20 0.40
HDAC1 Q13547 2/20 0.40
THRB P10828 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
GFER P55789 1/20 0.40
PLEC Q15149 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ERAP2 Q6P179 1/20 0.39
LNPEP Q9UIQ6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17336829 0.88 ALOX15 (0.58) ALOX15AAK1CYP17A1PRKCIMAPT
SCHEMBL29446496 0.88 ALOX15 (0.58) ALOX15AAK1CYP17A1PRKCIMAPT
SCHEMBL14876842 0.88 GAA (0.54) ALOX15AAK1CYP17A1PRKCIMAPT
SCHEMBL4516629 0.87 MAPT (0.55) ALOX15AAK1CYP17A1MAPTGAA
SCHEMBL21648056 0.86 ALOX15 (0.44) ALOX15AAK1CYP17A1PRKCIMAPT
SCHEMBL25254382 0.86 CSF1R (0.46) AAK1CYP17A1HDAC1
SCHEMBL5869074 0.83 ABCC9 (0.48) ALOX15AAK1CYP17A1MAPTGAA
SCHEMBL3410364 0.83 HPGD (0.49) ALOX15AAK1CYP17A1ALDH1A1HPGD
SCHEMBL15160030 0.83 GAA (0.52) ALOX15AAK1CYP17A1MAPTGAA
SCHEMBL753526 0.82 PTGER4 (0.57) ALOX15AAK1GAAERAP2LNPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113461602-B Aniline compounds with HDAC (Histone deacetylase) inhibitory activity, preparation method, composition and application 北京华氏信华科生物科技有限公司 2022-06-28 CN disclosed
CN-113461602-A Aniline compounds with HDAC (HDAC) inhibitory activity, preparation method, composition and application 北京华氏信华科生物科技有限公司 2021-10-01 CN disclosed