SCHEMBL28629150

SCHEMBL28629150

COc1ccc(OC(F)(F)F)cc1CCBr

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.49
TAAR1 Q96RJ0 1/20 0.49
AOC3 Q16853 1/20 0.44
HCRTR1 O43613 1/20 0.44
HCRTR2 O43614 1/20 0.44
TACR1 P25103 7/20 0.42
KCNH2 Q12809 2/20 0.42
CYP2D6 P10635 1/20 0.42
GRIN2B Q13224 2/20 0.42
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HRH1 P35367 1/20 0.42
HTR2B P41595 1/20 0.42
SLC6A3 Q01959 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3202940 0.87 TACR1 (0.46) ADRA1ATAAR1HCRTR1HCRTR2TACR1
SCHEMBL28620798 0.84 ADRA1A (0.49) ADRA1ATAAR1AOC3HCRTR1HCRTR2
SCHEMBL31284962 0.84 TAAR1 (0.71) ADRA1ATAAR1AOC3HCRTR1HCRTR2
SCHEMBL25308876 0.83 ADRA1A (0.68) ADRA1ATAAR1AOC3HTR2AHTR2C
SCHEMBL22220774 0.82 HCRTR1 (0.49) ADRA1ATAAR1HCRTR1HCRTR2TACR1
SCHEMBL4638450 0.81 GRIN2B (0.46) ADRA1ATAAR1HCRTR1HCRTR2TACR1
SCHEMBL15173398 0.81 ADRA1A (0.51) ADRA1ATAAR1AOC3HCRTR1HCRTR2
SCHEMBL3205585 0.81 HCRTR1 (0.46) ADRA1ATAAR1HCRTR1HCRTR2TACR1
SCHEMBL16892229 0.81 IDO1 (0.51) ADRA1ATAAR1HCRTR1HCRTR2TACR1
SCHEMBL27778188 0.79 GPR3 (0.40) AOC3SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108395396-B Preparation method of chiral o-amino alcohol intermediate, antagonist and analogue thereof 复旦大学 2021-07-23 CN disclosed