SCHEMBL28629620

SCHEMBL28629620

O=C(O)CCCc1cc(I)ccc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F13A1 P00488 3/20 0.43
HDAC3 O15379 1/20 0.42
MAPK1 P28482 1/20 0.42
ADRA1A P35348 1/20 0.42
HDAC4 P56524 1/20 0.42
SLC6A3 Q01959 1/20 0.42
HDAC1 Q13547 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
FFAR1 O14842 2/20 0.40
FFAR4 Q5NUL3 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8240809 0.83 PSEN1 (0.47) F13A1HDAC3MAPK1ADRA1AHDAC4
SCHEMBL6686448 0.81 FFAR4 (0.51) F13A1HDAC3MAPK1ADRA1AHDAC4
SCHEMBL19584858 0.80 NPC1 (0.45) F13A1HDAC3MAPK1ADRA1AHDAC4
SCHEMBL31018263 0.79 FFAR1 (0.56) FFAR1FFAR4GPR17AKR1B1
SCHEMBL29126694 0.78 NPSR1 (0.52) F13A1HDAC3MAPK1ADRA1AHDAC4
SCHEMBL29126688 0.78 IDO1 (0.45) F13A1HDAC3MAPK1ADRA1AHDAC4
SCHEMBL8239860 0.78 F13A1 (0.53) F13A1FFAR1FFAR4
SCHEMBL30428070 0.78 F13A1 (0.41) F13A1HDAC3MAPK1ADRA1AHDAC4
SCHEMBL29009780 0.78 MGLL (0.47) F13A1FFAR1FFAR4
SCHEMBL29009842 0.78 F13A1 (0.41) F13A1HDAC3MAPK1ADRA1AHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109608464-B Radioiodine-labeled Larotrectinib compound and preparation method and application thereof 上海健康医学院 2021-09-24 CN disclosed