SCHEMBL28630174

SCHEMBL28630174

COC(=O)C1(c2cccn2Cc2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.46
BRD2 P25440 1/20 0.46
BRD3 Q15059 1/20 0.46
BRDT Q58F21 1/20 0.46
TP53 P04637 1/20 0.46
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
OPRD1 P41143 1/20 0.43
CACNA1G O43497 1/20 0.42
CACNA1H O95180 1/20 0.42
CACNA1I Q9P0X4 1/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ADRA1D P25100 1/20 0.42
NOTUM Q6P988 1/20 0.41
CNR2 P34972 3/20 0.41
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25433106 0.74 SCD (0.47) ALDH1A1CACNA1GCACNA1HCACNA1IMAPT
SCHEMBL6746046 0.72 KDM4E (0.60) KDM4EALDH1A1POLBOPRD1ADRA1D
SCHEMBL1243976 0.72 CNR2 (0.55) BRD4BRD2BRD3BRDTTP53
SCHEMBL26637780 0.71 GAA (0.49) KDM4EALDH1A1POLBOPRD1ADRA1D
SCHEMBL10965858 0.71 BRD4 (0.50) BRD4BRD2BRD3BRDTTP53
SCHEMBL17042553 0.70 CYP2D6 (0.55) ALDH1A1MEN1KMT2ACYP2C9CYP2C19
SCHEMBL10567213 0.70 OPRM1 (0.53) KDM4EALDH1A1POLBOPRD1ADRA1D
SCHEMBL25433618 0.70 HDAC9 (0.43) TP53ALDH1A1LMNACACNA1GCACNA1H
SCHEMBL349195 0.70 MEN1 (0.56) OPRD1MEN1KMT2A
SCHEMBL8503086 0.70 CA12 (0.57) BRD4BRD2BRD3BRDTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693701-B Modulators of ATP-binding cassette transporters 弗特克斯药品有限公司 2021-08-10 CN disclosed