SCHEMBL28630958

SCHEMBL28630958

COC(=O)c1cc(-c2cccnc2)oc1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.50
CFTR P13569 1/20 0.49
SLC2A1 P11166 1/20 0.49
CYP19A1 P11511 1/20 0.49
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
ALDH1A1 P00352 2/20 0.48
EDNRA P25101 1/20 0.47
MAPK1 P28482 1/20 0.47
LMNA P02545 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
GABRA1 P14867 1/20 0.45
GABRG2 P18507 1/20 0.45
GABRB3 P28472 1/20 0.45
GABRA3 P34903 1/20 0.45
GABRA2 P47869 1/20 0.45
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24951908 0.85 NPC1 (0.56) ALDH1A1MAPK1LMNASMN1; SMN2HPGD
SCHEMBL29742813 0.85 NPC1 (0.56) ALDH1A1MAPK1LMNASMN1; SMN2HPGD
SCHEMBL29742828 0.83 MKNK1 (0.45) ALDH1A1LMNAMAPTHPGDKMT2A
SCHEMBL24951909 0.83 MKNK1 (0.45) ALDH1A1LMNAMAPTHPGDKMT2A
SCHEMBL2665747 0.83 ALDH1A1 (0.61) ALDH1A1MAPK1LMNASMN1; SMN2MAPT
SCHEMBL12876531 0.79 ALDH1A1 (0.48) ALDH1A1EDNRAMAPK1LMNASMN1; SMN2
SCHEMBL3101392 0.77 HDAC6 (0.52) ALDH1A1MAPK1SMN1; SMN2MAPTHPGD
SCHEMBL4184070 0.77 ALDH1A1 (0.44) ALDH1A1EDNRAMAPK1LMNASMN1; SMN2
SCHEMBL3107571 0.77 NPC1 (0.44) ALDH1A1EDNRAMAPK1SMN1; SMN2MAPT
SCHEMBL17212160 0.77 ALDH1A1 (0.53) NR4A2CYP19A1CYP11B1CYP11B2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113444081-B Thiadiazole carboxamide compounds and application thereof 浙江大学 2022-07-05 CN disclosed
CN-113444081-A Thiadiazole amide compound and application thereof 浙江大学 2021-09-28 CN disclosed