SCHEMBL28633277

SCHEMBL28633277

[CH2]c1ccc(/C=C/C(=O)Nc2ccccc2N)cc1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 17/20 0.63
HDAC2 Q92769 4/20 0.59
MMP1 P03956 3/20 0.56
MMP2 P08253 3/20 0.56
MMP9 P14780 3/20 0.56
EGFR P00533 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2640602 0.88 HDAC1 (0.66) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL3228591 0.88 EGFR (0.71) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL3228583 0.88 EGFR (0.71) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL7978520 0.87 HDAC1 (0.64) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL8348482 0.85 TRPA1 (0.68) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL4536420 0.85 TRPA1 (0.68) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL4536422 0.85 TRPA1 (0.68) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL13180844 0.85 HDAC1 (0.74) HDAC1HDAC2MMP1MMP2MMP9
SCHEMBL1064700 0.84 HDAC1 (0.65) HDAC1HDAC2
SCHEMBL1064701 0.84 HDAC1 (0.65) HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153636-B Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors 朱比连特埃皮科尔有限责任公司 2021-10-22 CN disclosed