SCHEMBL28633834

SCHEMBL28633834

COc1cc2c(cc1Br)CCCC2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.50
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
HTR2B P41595 1/20 0.49
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TSHR P16473 1/20 0.44
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAOA P21397 2/20 0.42
MAOB P27338 2/20 0.42
PRKCI P41743 1/20 0.42
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14052726 0.93 HSD17B1 (0.50) HSD17B1HTR2AHTR2CHTR2BMEN1
SCHEMBL30759603 0.93 HSD17B1 (0.50) HSD17B1HTR2AHTR2CHTR2BMEN1
SCHEMBL24362699 0.90 HTR2A (0.49) HSD17B1HTR2AHTR2CHTR2BMEN1
SCHEMBL1561740 0.89 HTR2A (0.51) HTR2AHTR2CHTR2BMEN1KMT2A
SCHEMBL424613 0.87 HSD17B1 (0.54) HSD17B1MEN1KMT2AMAPK1NPSR1
SCHEMBL9621112 0.84 KMT2A (0.53) HSD17B1MEN1KMT2AMAPK1NPSR1
SCHEMBL9621080 0.84 KMT2A (0.53) HSD17B1MEN1KMT2AMAPK1NPSR1
SCHEMBL2776025 0.83 HSD17B1 (0.50) HSD17B1MEN1KMT2AMAPK1NPSR1
SCHEMBL2306816 0.82 HTR2A (0.51) HTR2AHTR2CHTR2BMEN1KMT2A
SCHEMBL30759612 0.82 HTR2A (0.51) HTR2AHTR2CHTR2BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed