SCHEMBL9621080

SCHEMBL9621080

COc1cc2c(cc1OC)C(=O)CCCCC2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
MEN1 O00255 2/20 0.53
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 5/20 0.50
HSD17B1 P14061 1/20 0.50
CYP3A4 P08684 2/20 0.49
MAPT P10636 4/20 0.47
ACHE P22303 1/20 0.47
GAA P10253 1/20 0.47
MAOA P21397 1/20 0.47
HSD17B10 Q99714 2/20 0.47
MAPK1 P28482 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HPGD P15428 2/20 0.45
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.45
CYP19A1 P11511 1/20 0.44
CYP11B2 P19099 1/20 0.44
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9621112 1.00 KMT2A (0.53) KMT2AMEN1KDM4EALDH1A1HSD17B1
SCHEMBL424613 0.96 HSD17B1 (0.54) KMT2AMEN1KDM4EALDH1A1HSD17B1
SCHEMBL29420327 0.88 KMT2A (0.56) KMT2AMEN1KDM4EALDH1A1CYP3A4
SCHEMBL29420326 0.88 KMT2A (0.56) KMT2AMEN1KDM4EALDH1A1CYP3A4
SCHEMBL354177 0.88 KMT2A (0.56) KMT2AMEN1KDM4EALDH1A1CYP3A4
SCHEMBL24362699 0.87 HTR2A (0.49) KMT2AMEN1KDM4EHSD17B1CYP3A4
SCHEMBL24362549 0.87 HSD17B1 (0.47) KMT2AMEN1KDM4EALDH1A1HSD17B1
SCHEMBL25369104 0.86 HSD17B1 (0.46) KMT2AMEN1KDM4EALDH1A1HSD17B1
SCHEMBL24362546 0.86 MAPK10 (0.46) KMT2AMEN1HSD17B1MAPTMAOA
SCHEMBL9620643 0.86 ACHE (0.54) HSD17B1ACHEMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284359-B1 1,4-DISUBSTITUTED PIPERAZINE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-01-08 EP disclosed
US-4880809-A HYPOTENSIVE AGENTS, AMIDE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-11-14 US disclosed