SCHEMBL28634299

SCHEMBL28634299

COc1cc(-c2cccc(C(C)C)c2CC(N)=O)ccn1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 6/20 0.44
PKN1 Q16512 1/20 0.42
PKN2 Q16513 1/20 0.42
IDO1 P14902 1/20 0.39
LPAR1 Q92633 1/20 0.39
CNR1 P21554 1/20 0.39
WNT3A P56704 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
CYP3A4 P08684 1/20 0.38
SYK P43405 1/20 0.38
ACVR2A P27037 1/20 0.38
TGFBR2 P37173 1/20 0.38
PDE4B Q07343 1/20 0.37
PDE7A Q13946 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
AAK1 Q2M2I8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21962143 0.90 NLRP3 (0.45) NLRP3PKN1PKN2IDO1LPAR1
SCHEMBL21962099 0.89 NLRP3 (0.44) NLRP3PKN1PKN2IDO1LPAR1
SCHEMBL21962081 0.89 NLRP3 (0.46) NLRP3PKN1PKN2IDO1LPAR1
SCHEMBL22014327 0.83 NLRP3 (0.42) NLRP3IDO1ACVR2ATGFBR2PDE4B
SCHEMBL25067031 0.80 FFAR1 (0.39) NLRP3LPAR1WNT3A
SCHEMBL23063148 0.78 NLRP3 (0.45) NLRP3PKN1PKN2IDO1CNR1
SCHEMBL25144807 0.78 ACVR2A (0.43) NLRP3PKN1PKN2IDO1ACVR2A
SCHEMBL24787851 0.78 ACACB (0.40) NLRP3PKN2CDK5
SCHEMBL23012916 0.77 FFAR1 (0.37) NLRP3LPAR1WNT3A
SCHEMBL29691434 0.77 FFAR1 (0.37) NLRP3LPAR1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113227055-A Compounds and compositions for treating conditions associated with NLRP activity 诺华股份有限公司 2021-08-06 CN disclosed