SCHEMBL28634476

SCHEMBL28634476

COC(=O)c1csc(C(CC(N)C(C)C)O[Si](C)(C)C(C)(C)C)n1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 6/20 0.38
CA2 P00918 1/20 0.35
MAOA P21397 1/20 0.33
ACHE P22303 1/20 0.33
PTPRB P23467 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
TLR7 Q9NYK1 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28634475 1.00 ABCB1 (0.38) ABCB1CA2MAOAACHEPTPRB
SCHEMBL24140397 0.89 ABCB1 (0.48) ABCB1CA2PTPRBMEN1NPC1
SCHEMBL14765446 0.85 ABCB1 (0.38) ABCB1CA2MAOAACHEPTPRB
SCHEMBL19479759 0.82 ABCB1 (0.36) ABCB1CA2MAOAACHEMEN1
SCHEMBL28064131 0.82 ABCB1 (0.52) ABCB1CA2PTPRB
SCHEMBL28064130 0.82 ABCB1 (0.52) ABCB1CA2PTPRB
SCHEMBL17728762 0.80 ABCB1 (0.37) ABCB1CA2MAOAACHEMEN1
SCHEMBL22154581 0.80 ABCB1 (0.37) ABCB1CA2PTPRB
SCHEMBL28646527 0.80 ABCB1 (0.37) ABCB1CA2PTPRB
SCHEMBL19389074 0.79 ABCB1 (0.39) ABCB1CA2MAOAACHEPTPRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113454097-A Tubulysins and protein-tubulysin conjugates 里珍纳龙药品有限公司 2021-09-28 CN disclosed