SCHEMBL28634663

SCHEMBL28634663

COCCOc1cc(C(=O)O)cc(OC(F)F)n1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.36
HCAR3 P49019 3/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
PLA2G2A P14555 1/20 0.34
GCK P35557 3/20 0.34
ACACB O00763 2/20 0.34
RAF1 P04049 1/20 0.34
HTT P42858 1/20 0.33
RARG P13631 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30016380 1.00 FFAR4 (0.37) FFAR4MRGPRX4HCAR3ALDH1A1KDM4E
SCHEMBL28646014 0.89 KDM4E (0.50) FFAR4ALDH1A1KDM4EACACBRAF1
SCHEMBL28925140 0.82 MRGPRX4 (0.33) MRGPRX4PLA2G2ARAF1
SCHEMBL19330200 0.82 KDM4E (0.53) ALDH1A1KDM4EHTT
SCHEMBL30340556 0.82 KDM4E (0.53) ALDH1A1KDM4EHTT
SCHEMBL3714048 0.79 TAS1R3 (0.40) FFAR4HCAR3ALDH1A1KDM4EPLA2G2A
SCHEMBL30017038 0.77 TPMT (0.38) MRGPRX4ALDH1A1KDM4E
SCHEMBL21349298 0.77 TPMT (0.38) MRGPRX4ALDH1A1KDM4E
SCHEMBL89628 0.76 KDM4E (0.50) FFAR4HCAR3ALDH1A1KDM4EPLA2G2A
SCHEMBL2711725 0.75 KDM4E (0.46) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113264945-B Spiro derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113264945-A Spiro derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-08-17 CN disclosed