SCHEMBL28634741

SCHEMBL28634741

COc1nccc(S)c1Cl.[NaH]

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.35
CCR4 P51679 3/20 0.34
GPBAR1 Q8TDU6 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDCD1 Q15116 3/20 0.33
CD274 Q9NZQ7 3/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 1/20 0.33
APLNR P35414 1/20 0.33
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
AURKA O14965 1/20 0.32
TTK P33981 1/20 0.32
AURKB Q96GD4 1/20 0.32
INCENP Q9NQS7 1/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18328238 0.98 NFE2L2 (0.36) NFE2L2CCR4GPBAR1MAPK1L3MBTL1
SCHEMBL18328236 0.78 HPGD (0.46) MAPK1L3MBTL1CD274KMT2AALDH1A1
SCHEMBL188900 0.78 HPGD (0.36) NFE2L2CCR4GPBAR1MAPK1L3MBTL1
SCHEMBL911419 0.77 CCR4 (0.43) NFE2L2CCR4MAPK1L3MBTL1MAPT
SCHEMBL26026672 0.75 TRPA1 (0.35) NFE2L2MAPTKMT2AAPLNRCCR1
SCHEMBL5942324 0.75 DRD1 (0.39) NFE2L2CCR4GPBAR1MAPK1L3MBTL1
SCHEMBL27849554 0.75 MAPK1 (0.45) CCR4MAPK1L3MBTL1MAPTKMT2A
SCHEMBL21063375 0.73 CCR4 (0.35) NFE2L2CCR4GPBAR1MAPK1L3MBTL1
SCHEMBL21598410 0.73 CCR4 (0.37) NFE2L2CCR4GPBAR1MAPK1L3MBTL1
SCHEMBL21598414 0.73 AURKA (0.43) CCR4MAPK1L3MBTL1PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113272303-A Pyrimido five-membered nitrogen heterocyclic derivative, preparation method and application thereof in medicine 上海拓界生物医药科技有限公司 2021-08-17 CN disclosed