SCHEMBL28634847

SCHEMBL28634847

COc1cc(Cl)ncc1-c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 6/20 0.56
CYP11B2 P19099 6/20 0.56
CYP19A1 P11511 4/20 0.56
CYP17A1 P05093 3/20 0.56
MKNK1 Q9BUB5 2/20 0.53
MKNK2 Q9HBH9 2/20 0.53
CYP3A4 P08684 4/20 0.50
CYP2A6 P11509 2/20 0.50
PDE10A Q9Y233 1/20 0.50
PDGFRB P09619 1/20 0.49
PDGFRA P16234 1/20 0.49
MAPK1 P28482 2/20 0.48
POLB P06746 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HSD17B10 Q99714 1/20 0.48
HTT P42858 1/20 0.48
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ERN1 O75460 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28225240 0.79 MKNK1 (0.60) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL28018862 0.77 CYP11B1 (0.56) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL28118939 0.77 CYP11B1 (0.61) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL23326169 0.75 MKNK1 (0.56) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL29775379 0.75 MKNK1 (0.56) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL4506402 0.75 CYP11B1 (0.60) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL14680957 0.75 MKNK1 (0.63) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL12381484 0.74 CYP11B1 (0.74) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL31663902 0.74 MKNK1 (0.62) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1
SCHEMBL21076869 0.74 MKNK1 (0.66) CYP11B1CYP11B2CYP19A1CYP17A1MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113574055-A PCSK9 inhibitors and methods of use thereof 阿斯利康(瑞典)有限公司 2021-10-29 CN disclosed
CN-113412258-A PCSK9 inhibitors and methods of use thereof 阿斯利康(瑞典)有限公司 2021-09-17 CN disclosed