SCHEMBL28634877

SCHEMBL28634877

Cc1ccc(Cn2cnc3ccc(Br)cc3c2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.54
HDAC6 Q9UBN7 3/20 0.53
LMNA P02545 2/20 0.51
HDAC3 O15379 2/20 0.51
HDAC4 P56524 2/20 0.51
HDAC1 Q13547 2/20 0.51
HDAC7 Q8WUI4 2/20 0.51
HDAC2 Q92769 2/20 0.51
HDAC10 Q969S8 2/20 0.51
HDAC11 Q96DB2 2/20 0.51
HDAC8 Q9BY41 2/20 0.51
HDAC9 Q9UKV0 2/20 0.51
HDAC5 Q9UQL6 2/20 0.51
GRK2 P25098 1/20 0.50
TP53 P04637 1/20 0.49
DDR1 Q08345 1/20 0.48
SCD O00767 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30669835 1.00 MCL1 (0.54) MCL1HDAC6LMNAHDAC3HDAC4
SCHEMBL1500148 0.86 GRK2 (0.65) MCL1GRK2SCDMMP13
SCHEMBL29723994 0.86 GRK2 (0.65) MCL1GRK2SCDMMP13
SCHEMBL29147374 0.86 MMP13 (0.64) MCL1HDAC6LMNAHDAC3HDAC4
SCHEMBL2315222 0.82 GRK2 (0.50) MCL1HDAC6HDAC3HDAC4HDAC1
SCHEMBL29065789 0.81 GRK2 (0.65) GRK2TP53SMN1; SMN2MMP13TRPA1
SCHEMBL2611259 0.81 HDAC6 (0.67) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL5529666 0.81 SMN1; SMN2 (0.67) HDAC6LMNAHDAC1TP53SMN1; SMN2
SCHEMBL4210572 0.80 MCL1 (0.61) MCL1LMNADDR1SMN1; SMN2HTT
SCHEMBL2317430 0.80 SCD (0.63) HDAC6LMNAHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113461661-B 6- (pyridin-3-yl) quinazoline-4 (3H) -ketone derivative and preparation and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2023-11-28 CN disclosed
CN-113461661-A 6- (pyridine-3-yl) quinazoline-4 (3H) -ketone derivative and preparation and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2021-10-01 CN disclosed