SCHEMBL29147374

SCHEMBL29147374

COc1ccc(Cn2cnc3ccc(Br)cc3c2=O)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 5/20 0.64
MCL1 Q07820 1/20 0.54
LMNA P02545 1/20 0.54
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC2 Q92769 1/20 0.53
HDAC10 Q969S8 1/20 0.53
HDAC11 Q96DB2 1/20 0.53
HDAC8 Q9BY41 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
HDAC9 Q9UKV0 1/20 0.53
HDAC5 Q9UQL6 1/20 0.53
SLC22A8 Q8TCC7 1/20 0.52
GRK2 P25098 4/20 0.51
ROCK1 Q13464 2/20 0.51
AURKA O14965 1/20 0.51
PRKCB P05771 1/20 0.51
AKT1 P31749 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3085533 0.90 MMP13 (0.55) MMP13HDAC3HDAC4HDAC1HDAC7
SCHEMBL19338476 0.86 MMP13 (0.65) MMP13HDAC3HDAC4HDAC1HDAC7
SCHEMBL28634877 0.86 MCL1 (0.54) MMP13MCL1LMNAHDAC3HDAC4
SCHEMBL30669835 0.86 MCL1 (0.54) MMP13MCL1LMNAHDAC3HDAC4
SCHEMBL2491607 0.85 MMP13 (0.64) MMP13HDAC3HDAC4HDAC1HDAC7
SCHEMBL2315834 0.85 MMP13 (0.64) MMP13HDAC3HDAC4HDAC1HDAC7
SCHEMBL29723994 0.83 GRK2 (0.65) MMP13MCL1GRK2GRK5
SCHEMBL1500148 0.83 GRK2 (0.65) MMP13MCL1GRK2GRK5
SCHEMBL29433505 0.82 QPCT (0.58) MMP13LMNAMAPTTSHRKDM4E
SCHEMBL15825080 0.82 QPCT (0.58) MMP13LMNAMAPTTSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113501819-B Pyridoimidazole substituted quinazolinone derivative, and synthetic method and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2024-02-02 CN disclosed