SCHEMBL2863572

SCHEMBL2863572

CC[C@@H](N)c1ccc(C)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.46
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2E1 P05181 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
ADRA2A P08913 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
ROCK1 Q13464 1/20 0.35
ELANE P08246 1/20 0.34
P2RX7 Q99572 2/20 0.33
HRH1 P35367 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
MAPK1 P28482 1/20 0.32
ESR1 P03372 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2674305 1.00 SLC6A4 (0.46) SLC6A4MEN1LMNAKMT2ACYP1A2
Hydrochloric Acid SCHEMBL2749385 0.98 SLC6A4 (0.44) SLC6A4MEN1LMNAKMT2ACYP1A2
SCHEMBL20184239 0.82 ADRA2A (0.39) MEN1LMNAKMT2ACYP1A2CYP2E1
SCHEMBL2760888 0.82 ADRA2A (0.39) MEN1LMNAKMT2ACYP1A2CYP2E1
SCHEMBL14480428 0.82 ADRA2A (0.39) MEN1LMNAKMT2ACYP1A2CYP2E1
Hydrochloric Acid SCHEMBL1440347 0.81 ADRA2A (0.41) MEN1LMNAKMT2ACYP1A2CYP2E1
Hydrochloric Acid SCHEMBL1440350 0.81 ADRA2A (0.41) MEN1LMNAKMT2ACYP1A2CYP2E1
Hydrochloric Acid SCHEMBL1440719 0.81 ADRA2A (0.41) MEN1LMNAKMT2ACYP1A2CYP2E1
SCHEMBL998729 0.79 P2RX3 (0.37) MEN1LMNAKMT2ACYP1A2CYP2E1
SCHEMBL998728 0.79 P2RX3 (0.37) MEN1LMNAKMT2ACYP1A2CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139334-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2010-01-06 EP disclosed
EP-2136639-A1 PYRID-2-YL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2009-12-30 EP disclosed
WO-2008130481-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2008-10-30 WO disclosed
WO-2008123963-A1 PYRID-2-YL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2008-10-16 WO disclosed