SCHEMBL28636159

SCHEMBL28636159

CC(C)c1ccc(-c2nc(-c3ccc(C=O)cc3Cl)no2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 1/20 0.43
HSD11B1 P28845 1/20 0.43
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
S1PR1 P21453 4/20 0.39
S1PR3 Q99500 2/20 0.39
S1PR5 Q9H228 1/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28638941 0.86 S1PR1 (0.46) HSD11B1NPC1RAB9ASMN1; SMN2S1PR1
SCHEMBL4741601 0.86 S1PR1 (0.52) S1PR1S1PR3S1PR5MAP4K4MINK1
SCHEMBL28636374 0.85 RAB9A (0.49) NPC1RAB9AMEN1CYP1A2CYP2C19
SCHEMBL28636386 0.84 NPC1 (0.49) HSD11B1NPC1RAB9AMEN1CYP1A2
SCHEMBL28656533 0.84 S1PR1 (0.57) S1PR1S1PR3S1PR5MAP4K4MINK1
SCHEMBL19287102 0.83 TYR (0.56) TYRNPC1RAB9AMEN1CYP1A2
SCHEMBL28657010 0.80 S1PR1 (0.55) S1PR1S1PR3S1PR5
SCHEMBL28636371 0.80 MAOA (0.44) NPC1RAB9AMEN1CYP1A2CYP2C19
SCHEMBL1964923 0.78 S1PR1 (0.53) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL28638111 0.77 S1PR1 (0.57) S1PR1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109956912-B Carboxylic acid compound containing diphenyl oxadiazole, preparation method and medical application thereof 中国医学科学院药物研究所 2021-10-22 CN disclosed