SCHEMBL28636864

SCHEMBL28636864

CON(C)C(=O)c1ccccc1C(C)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.40
LMNA P02545 4/20 0.40
TP53 P04637 2/20 0.40
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 2/20 0.40
TRPM8 Q7Z2W7 1/20 0.39
MLYCD O95822 1/20 0.39
TSHR P16473 2/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 4/20 0.38
MEN1 O00255 1/20 0.38
CLK1 P49759 1/20 0.36
DYRK1A Q13627 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
CFTR P13569 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12347521 0.83 ALDH1A1 (0.44) SMN1; SMN2LMNATP53ALDH1A1KDM4E
SCHEMBL4611372 0.81 KMT2A (0.53) LMNATP53ALDH1A1TRPM8TSHR
SCHEMBL15938456 0.81 TSHR (0.55) SMN1; SMN2LMNAALDH1A1KDM4ETRPM8
SCHEMBL3309083 0.80 AKR1C3 (0.53) SMN1; SMN2LMNAALDH1A1KDM4ETSHR
SCHEMBL14164778 0.79 MEN1 (0.57) SMN1; SMN2LMNATP53ALDH1A1KDM4E
SCHEMBL308205 0.79 POLB (0.59) TP53ALDH1A1TSHRKMT2APOLB
SCHEMBL29215007 0.79 TSHR (0.60) SMN1; SMN2LMNATP53ALDH1A1KDM4E
SCHEMBL33252 0.79 ALDH1A1 (0.56) SMN1; SMN2TP53ALDH1A1KDM4ETRPM8
SCHEMBL306847 0.79 HPGD (0.54) SMN1; SMN2TP53ALDH1A1KDM4ETRPM8
SCHEMBL29898808 0.79 KMT2A (0.54) SMN1; SMN2ALDH1A1MLYCDGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549015-B Preparation method and application of 4-substituted phthalazinone derivative 安徽工业大学 2023-07-14 CN disclosed
CN-113549015-A Preparation method and application of 4-substituted phthalazinone derivative 安徽工业大学 2021-10-26 CN disclosed