SCHEMBL28637112

SCHEMBL28637112

CC(O)c1cccc(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GLS O94925 5/20 0.48
BRD4 O60885 3/20 0.45
KDM4A O75164 1/20 0.45
CREBBP Q92793 1/20 0.44
NAMPT P43490 2/20 0.43
CTSK P43235 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA7 P43166 1/20 0.42
CA14 Q9ULX7 1/20 0.42
SYK P43405 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21089822 1.00 GLS (0.48) GLSBRD4KDM4ACREBBPNAMPT
SCHEMBL12318659 0.90 GLS (0.49) GLSBRD4KDM4ACREBBPNAMPT
SCHEMBL27779357 0.88 GLS (0.47) GLSBRD4KDM4ACREBBPNAMPT
SCHEMBL13715120 0.86 GLS (0.46) GLSBRD4KDM4ACREBBPNAMPT
SCHEMBL14898071 0.85 GLS (0.48) GLSBRD4KDM4ACREBBPNAMPT
SCHEMBL25908751 0.84 GLS (0.51) GLSBRD4KDM4ACREBBPNAMPT
SCHEMBL23413688 0.83 GLS (0.46) GLSBRD4KDM4ACREBBPCTSK
SCHEMBL31389110 0.82 SYK (0.46) GLSBRD4KDM4ACREBBPNAMPT
SCHEMBL30771369 0.81 SYK (0.46) GLSBRD4KDM4ACREBBPNAMPT
SCHEMBL7865716 0.81 GLS (0.49) GLSBRD4KDM4ACREBBPNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689661-B Macrocyclic inhibitors of myeloperoxidase 百时美施贵宝公司 2021-10-15 CN disclosed