SCHEMBL28637731

SCHEMBL28637731

COC(=O)c1ccc(CN(C(=O)N2CCSCC2)c2ccc(F)cc2)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 4/20 0.39
PTGER2 P43116 1/20 0.38
CXCR2 P25025 2/20 0.37
MAPK1 P28482 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
STAT3 P40763 1/20 0.36
MLYCD O95822 2/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CXCR1 P25024 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28643589 0.90 MAPK1 (0.36) MAPK1KMT2ANPC1RAB9ASTAT3
SCHEMBL28634554 0.90 HSD17B10 (0.39) MAPK1KMT2ANPC1RAB9AMEN1
SCHEMBL28627863 0.90 ALDH1A1 (0.42) GABRA5MAPK1KMT2ANPC1RAB9A
SCHEMBL22218222 0.89 KMT2A (0.38) GABRA5PTGER2CXCR2MAPK1KMT2A
SCHEMBL28634587 0.89 HDAC1 (0.43) GABRA5HDAC1HDAC8HDAC6HDAC5
SCHEMBL20236480 0.88 HRH3 (0.41) GABRA5PTGER2CXCR2MAPK1KMT2A
SCHEMBL22218015 0.88 HRH3 (0.46) CXCR2KMT2AMEN1HRH3KDM4E
SCHEMBL22218289 0.88 MLYCD (0.46) GABRA5KMT2AMEN1MLYCDHRH3
SCHEMBL22217975 0.87 ALDH1A1 (0.41) GABRA5PTGER2CXCR2MAPK1KMT2A
Hydrochloric Acid SCHEMBL20236387 0.87 HRH3 (0.41) GABRA5PTGER2CXCR2MAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137518-B 1,3, 4-oxadiazole derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same 株式会社钟根堂 2021-08-31 CN disclosed