SCHEMBL28637820

SCHEMBL28637820

CNc1cc(OC(C)C)cc(C2CC2)c1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.32
F2 P00734 2/20 0.32
PLG P00747 2/20 0.32
PLAU P00749 2/20 0.32
PLAT P00750 2/20 0.32
KLKB1 P03952 2/20 0.32
PRSS1 P07477 2/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
DRD4 P21917 1/20 0.31
HTR1A P08908 1/20 0.31
POLB P06746 1/20 0.31
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ABL1 P00519 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28642986 0.80 SLC18A3 (0.36) TSHRPOLB
SCHEMBL23793815 0.77 TSHR (0.34) TSHRPLGPLAUPLATKDM4E
SCHEMBL28926824 0.77 CNR2 (0.34) KDM4EALDH1A1NPC1HPGDRAB9A
SCHEMBL25484300 0.76 TSHR (0.33) TSHRPOLB
SCHEMBL28645681 0.75 DHODH (0.34)
SCHEMBL25494208 0.73 TSHR (0.32) TSHRPOLB
SCHEMBL26034932 0.73 GRIN2D (0.37) TSHRKDM4EALDH1A1HTR1APOLB
SCHEMBL25495087 0.73 TSHR (0.32) TSHRPOLB
SCHEMBL22090081 0.72 GRIN2D (0.40) TSHRPLGPLAUPLATKDM4E
SCHEMBL22089827 0.72 ALDH1A3 (0.47) TSHRALDH1A1POLBNPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113412113-B Amino oxazinamides 豪夫迈·罗氏有限公司 2024-07-26 CN disclosed
CN-113412113-A Aminooxazine amides 豪夫迈·罗氏有限公司 2021-09-17 CN disclosed