SCHEMBL28638256

SCHEMBL28638256

COCC(C)n1nc(-c2sc(N)nc2-c2ccc(F)cc2)ccc1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 3/20 0.43
FBP1 P09467 2/20 0.38
ADORA2A P29274 3/20 0.37
ADORA1 P30542 3/20 0.37
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
XBP1 P17861 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KCNH2 Q12809 1/20 0.35
EGFR P00533 1/20 0.34
MYC P01106 1/20 0.34
WDR5 P61964 1/20 0.34
ADORA2B P29275 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
TGFBR2 P37173 1/20 0.33
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6134033 0.86 TGFBR1 (0.48) TGFBR1FBP1ADORA2AADORA1KDM4E
SCHEMBL28640612 0.82 ADORA2A (0.47) TGFBR1FBP1ADORA2AADORA1KDM4E
SCHEMBL6134226 0.75 ALDH1A1 (0.51) TGFBR1FBP1KDM4EMAPTLMNA
SCHEMBL6133824 0.74 MAPT (0.39) TGFBR1FBP1ADORA2AADORA1KDM4E
Bromide SCHEMBL6133333 0.74 ALDH1A1 (0.50) TGFBR1FBP1KDM4EMAPTLMNA
SCHEMBL6134790 0.74 TGFBR1 (0.41) TGFBR1ADORA2AADORA1KDM4ESMN1; SMN2
SCHEMBL28647146 0.72 TGFBR1 (0.47) TGFBR1FBP1ADORA2AADORA1KDM4E
SCHEMBL6133930 0.72 RET (0.42) TGFBR1ADORA2AADORA1KDM4ETGFBR2
SCHEMBL28646803 0.72 ADORA2A (0.61) TGFBR1FBP1ADORA2AADORA1KDM4E
SCHEMBL6133042 0.71 ALDH1A1 (0.46) FBP1KDM4EMAPTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109293652-B Substituted thiazole derivative and application thereof 四川科伦博泰生物医药股份有限公司 2021-10-22 CN disclosed