SCHEMBL28638636

SCHEMBL28638636

O=Cc1cc(Br)c2cc[nH]c2c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.50
RHEB Q15382 1/20 0.46
AHR P35869 3/20 0.46
CSNK2A1 P68400 1/20 0.38
KIF11 P52732 2/20 0.36
ALDH1A1 P00352 3/20 0.34
PARP1 P09874 1/20 0.34
ALDH1A3 P47895 2/20 0.34
NR4A2 P43354 1/20 0.33
HTR6 P50406 1/20 0.33
ALDH3A1 P30838 1/20 0.33
CDK8 P49336 1/20 0.32
PRKCI P41743 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29954569 0.79 CYP2A6 (0.52) CYP2A6KIF11ALDH1A1ALDH1A3
SCHEMBL15652269 0.78 CYP2A6 (0.50) CYP2A6AHRKIF11ALDH1A1CDK8
SCHEMBL19586691 0.74 CYP2A6 (0.50) CYP2A6KIF11ALDH1A1ALDH1A3ALDH3A1
SCHEMBL29644241 0.74 AHR (0.54) CYP2A6RHEBAHRCSNK2A1ALDH1A1
SCHEMBL1020056 0.74 AHR (0.54) CYP2A6RHEBAHRCSNK2A1ALDH1A1
SCHEMBL16452861 0.74 ALDH1A1 (0.49) CYP2A6ALDH1A1ALDH1A3
SCHEMBL15475106 0.73 XDH (0.46) CYP2A6KIF11ALDH1A1ALDH1A3ALDH3A1
SCHEMBL2516555 0.71 RHEB (0.50) CYP2A6RHEBAHRCSNK2A1ALDH1A1
SCHEMBL996179 0.71 AHR (0.50) CYP2A6RHEBAHRCSNK2A1ALDH1A1
SCHEMBL31435859 0.71 RHEB (0.50) CYP2A6RHEBAHRCSNK2A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300129-B Heterocyclic compounds as BCR-ABL inhibitors 苏州亚盛药业有限公司 2021-09-14 CN disclosed