SCHEMBL28638657

SCHEMBL28638657

CNC(C)CCn1c(=O)c(-c2cccc(F)c2Cl)cn(CC(=O)OC)c1=O

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 15/20 0.41
CYP3A4 P08684 10/20 0.39
P2RX3 P56373 2/20 0.34
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28638656 0.84 GNRHR (0.41) GNRHRCYP3A4PDCD1CD274EGFR
SCHEMBL28651462 0.84 GNRHR (0.41) GNRHRCYP3A4PDCD1CD274EGFR
SCHEMBL28644101 0.82 GNRHR (0.40) GNRHRCYP3A4P2RX3PDCD1CD274
SCHEMBL28645661 0.82 GNRHR (0.40) GNRHRCYP3A4PDCD1CD274EGFR
SCHEMBL28638881 0.82 GNRHR (0.40) GNRHRCYP3A4PDCD1CD274EGFR
SCHEMBL28644084 0.81 GNRHR (0.39) GNRHRCYP3A4PDCD1CD274
SCHEMBL30178388 0.81 GNRHR (0.39) GNRHRCYP3A4PDCD1CD274EGFR
SCHEMBL28660744 0.79 GNRHR (0.40) GNRHRCYP3A4
SCHEMBL28663476 0.78 GNRHR (0.39) GNRHRCYP3A4P2RX3PDCD1CD274
SCHEMBL28663474 0.78 GNRHR (0.39) GNRHRCYP3A4P2RX3PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428744-B Novel heterocyclic compounds and their use in medicine and cosmetics 盖尔德马研究及发展公司 2021-09-24 CN disclosed