SCHEMBL28639031

SCHEMBL28639031

CCOC(=O)c1cc2c(cc1OCC)C(=O)N(Cc1ccccc1)C2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.57
MEN1 O00255 1/20 0.57
CASP3 P42574 1/20 0.51
TSHR P16473 1/20 0.46
HDAC4 P56524 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
PARP1 P09874 1/20 0.42
TRPC5 Q9UL62 1/20 0.42
HSP90AA1 P07900 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
TDP2 O95551 1/20 0.41
NSD2 O96028 1/20 0.41
PLCG1 P19174 1/20 0.41
PAX8 Q06710 1/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28638165 0.92 MEN1 (0.57) KMT2AMEN1CASP3TSHRHDAC4
SCHEMBL28633462 0.90 KMT2A (0.53) KMT2AMEN1CASP3HDAC4HDAC1
SCHEMBL28645766 0.90 MEN1 (0.53) KMT2AMEN1CASP3TSHRALDH1A1
SCHEMBL28925117 0.90 MEN1 (0.50) KMT2AMEN1CASP3HDAC4HDAC1
SCHEMBL28656587 0.90 TSHR (0.51) KMT2AMEN1CASP3TSHRPARP1
SCHEMBL30604585 0.90 MEN1 (0.47) KMT2AMEN1CASP3TSHRTRPC5
SCHEMBL30604599 0.90 MEN1 (0.53) KMT2AMEN1CASP3TSHRALDH1A1
SCHEMBL28633459 0.90 MEN1 (0.47) KMT2AMEN1CASP3TSHRTRPC5
SCHEMBL28645349 0.89 KMT2A (0.53) KMT2AMEN1CASP3HDAC1HSP90AA1
SCHEMBL30604582 0.89 KMT2A (0.53) KMT2AMEN1CASP3HDAC1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed