SCHEMBL28633459

SCHEMBL28633459

CCOC(=O)c1cc2c(cc1OCC)C(=O)N(Cc1ccccc1)CC2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
GRM5 P41594 1/20 0.47
TSHR P16473 1/20 0.45
CASP3 P42574 1/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
LMNA P02545 4/20 0.44
PKM P14618 2/20 0.44
MAPT P10636 1/20 0.43
ALDH1A1 P00352 4/20 0.43
TRPC5 Q9UL62 1/20 0.43
KCNK3 O14649 1/20 0.43
HTT P42858 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
AOC3 Q16853 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30604585 1.00 MEN1 (0.47) MEN1KMT2AGRM5TSHRCASP3
SCHEMBL28636452 0.91 KMT2A (0.51) MEN1KMT2AGRM5SMN1; SMN2LMNA
SCHEMBL30604607 0.91 KMT2A (0.51) MEN1KMT2AGRM5SMN1; SMN2LMNA
SCHEMBL28639031 0.90 KMT2A (0.57) MEN1KMT2ATSHRCASP3ALDH1A1
SCHEMBL28638924 0.83 GRM5 (0.52) MEN1KMT2AGRM5TSHRSMN1; SMN2
SCHEMBL30604584 0.83 GRM5 (0.52) MEN1KMT2AGRM5TSHRSMN1; SMN2
SCHEMBL28656587 0.82 TSHR (0.51) MEN1KMT2ATSHRCASP3SMN1; SMN2
SCHEMBL28638165 0.81 MEN1 (0.57) MEN1KMT2ATSHRCASP3SMN1; SMN2
SCHEMBL28633462 0.80 KMT2A (0.53) MEN1KMT2ACASP3MAPT
SCHEMBL30604599 0.80 MEN1 (0.53) MEN1KMT2ATSHRCASP3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed