SCHEMBL28633462

SCHEMBL28633462

CCOc1cc2c(cc1C(=O)O)CN(Cc1ccccc1)C2=O

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.49
HDAC1 Q13547 3/20 0.46
HDAC4 P56524 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
PARP1 P09874 1/20 0.45
CASP3 P42574 1/20 0.43
PREP P48147 1/20 0.42
HDAC7 Q8WUI4 1/20 0.41
USP2 O75604 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ALOX15 P16050 1/20 0.40
DHPS P49366 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28638917 0.90 KMT2A (0.47) KMT2AMEN1TDP1
SCHEMBL30604612 0.90 KMT2A (0.47) KMT2AMEN1TDP1
SCHEMBL30604606 0.90 KMT2A (0.45) KMT2AMEN1HDAC1HDAC4HDAC6
SCHEMBL28656930 0.90 KMT2A (0.45) KMT2AMEN1HDAC1HDAC4HDAC6
SCHEMBL28639031 0.90 KMT2A (0.57) KMT2AMEN1HDAC1HDAC4HDAC6
SCHEMBL28652153 0.90 KMT2A (0.53) KMT2AMEN1HDAC1HDAC4HDAC6
SCHEMBL30604571 0.90 KMT2A (0.53) KMT2AMEN1HDAC1HDAC4HDAC6
SCHEMBL30604607 0.89 KMT2A (0.51) KMT2AMEN1MAPTDHPS
SCHEMBL28636452 0.89 KMT2A (0.51) KMT2AMEN1MAPTDHPS
SCHEMBL28647745 0.88 HDAC1 (0.47) KMT2AMEN1HDAC1HDAC4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
CN-113493438-A Tetrahydroisoquinoline compounds 江苏先声药业有限公司 2021-10-12 CN disclosed