SCHEMBL28639683

SCHEMBL28639683

O=S(=O)(Nc1cccc(-c2nnn[nH]2)c1)c1ccc(-c2cccc(Cl)c2Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 9/20 0.49
LNPEP Q9UIQ6 1/20 0.47
GAA P10253 1/20 0.43
PFKFB4 Q16877 3/20 0.42
CYP19A1 P11511 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP8 P22894 1/20 0.42
MMP13 P45452 1/20 0.42
PTGES2 Q9H7Z7 1/20 0.41
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.38
PKM P14618 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL793726 0.85 PFKFB3 (0.67) PFKFB3LNPEPGAAPFKFB4CYP19A1
SCHEMBL794304 0.84 PFKFB3 (0.63) PFKFB3LNPEPPFKFB4MMP2MMP9
SCHEMBL793409 0.84 PFKFB3 (0.55) PFKFB3LNPEPPTGES2MEN1KMT2A
SCHEMBL27943370 0.82 MMP2 (0.59) PFKFB3GAAPFKFB4MMP2MMP9
SCHEMBL794544 0.81 PFKFB3 (0.59) PFKFB3LNPEPPFKFB4MMP2MMP9
SCHEMBL793555 0.81 PFKFB3 (0.66) PFKFB3LNPEPPFKFB4MEN1KMT2A
SCHEMBL793332 0.80 PFKFB3 (0.55) PFKFB3LNPEPGAAPFKFB4CYP19A1
SCHEMBL793433 0.79 PFKFB4 (0.67) PFKFB3PFKFB4CYP19A1PKM
SCHEMBL794311 0.78 PFKFB3 (0.65) PFKFB3LNPEPPFKFB4MEN1KMT2A
SCHEMBL794222 0.78 PFKFB3 (0.56) PFKFB3LNPEPGAAPFKFB4CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396145-A PFKFB3 inhibitors and uses thereof 盖罗发现有限责任公司 2021-09-14 CN disclosed