SCHEMBL28640545

SCHEMBL28640545

[CH2]C(=O)NNC(=S)Nc1cccc2ccccc12

nearest known ligand 0.75

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.75
GAA P10253 4/20 0.75
MAPT P10636 4/20 0.60
KMT2A Q03164 4/20 0.60
MEN1 O00255 3/20 0.60
ALOX12 P18054 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
ALPL P05186 1/20 0.59
KDM4E B2RXH2 6/20 0.56
RAB9A P51151 3/20 0.51
NPC1 O15118 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
POLB P06746 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19277764 0.84 GAA (0.75) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL4765694 0.81 KDM4E (0.69) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL1275812 0.81 KMT2A (0.72) ALDH1A1GAAKMT2AMEN1KDM4E
SCHEMBL6130342 0.80 ALDH1A1 (0.68) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL28220669 0.79 GAA (0.71) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL28182829 0.79 ALDH1A1 (0.66) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL28634224 0.78 EPHX1 (0.61) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL28635155 0.78 ALDH1A1 (0.59) ALDH1A1MAPTKMT2AMEN1ALOX12
SCHEMBL28645469 0.78 NPC1 (0.68) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL28638817 0.78 NPC1 (0.54) ALDH1A1GAAKMT2AMEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113480524-A Alkaloid hamacanthins series derivatives, and preparation method and application thereof 河北工业大学 2021-10-08 CN claimed
CN-113480524-B Alkaloid hamacanthins series derivatives, and preparation method and application thereof 河北工业大学 2022-08-30 CN disclosed
CN-113480524-A Alkaloid hamacanthins series derivatives, and preparation method and application thereof 河北工业大学 2021-10-08 CN disclosed