SCHEMBL28642575

SCHEMBL28642575

COC(=O)c1ccccc1-n1cncn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
MYC P01106 1/20 0.53
KMT2A Q03164 2/20 0.50
POLB P06746 4/20 0.49
HCRTR1 O43613 1/20 0.47
HCRTR2 O43614 1/20 0.47
KDM4E B2RXH2 3/20 0.45
TSHR P16473 2/20 0.45
LMNA P02545 1/20 0.45
ALDH1A1 P00352 3/20 0.44
HSD17B10 Q99714 2/20 0.44
CFTR P13569 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
ATM Q13315 1/20 0.42
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27314680 0.83 HCRTR1 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL30982330 0.81 HCRTR1 (0.51) CYP1A2CYP3A4CYP2C9CYP2C19MYC
SCHEMBL299870 0.81 HCRTR1 (0.48) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL403908 0.81 HCRTR1 (0.51) CYP1A2CYP3A4CYP2C9CYP2C19MYC
SCHEMBL28396855 0.80 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL10475608 0.79 KMT2A (0.51) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL19979962 0.78 CYP1A2 (0.46) CYP1A2CYP3A4CYP2C9CYP2C19POLB
SCHEMBL28397648 0.77 POLB (0.51) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL8193680 0.77 CYP1A2 (0.54) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL27787386 0.77 MYC (0.54) MYCKMT2APOLBHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113444016-A Molecules having pesticidal utility, and intermediates, compositions and methods related thereto 美国陶氏益农公司 2021-09-28 CN disclosed