SCHEMBL28397648

SCHEMBL28397648

COC(=O)c1cccc(Br)c1-n1cncn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.51
KDM4E B2RXH2 3/20 0.47
CYP1A2 P05177 3/20 0.45
CYP2C19 P33261 3/20 0.45
CYP2C9 P11712 2/20 0.45
CYP3A4 P08684 1/20 0.45
KMT2A Q03164 4/20 0.44
MEN1 O00255 2/20 0.44
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
SLC6A3 Q01959 1/20 0.37
MAPT P10636 3/20 0.36
CFTR P13569 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA5A P35218 1/20 0.36
CA9 Q16790 1/20 0.36
PTPRC P08575 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28642575 0.77 CYP1A2 (0.56) POLBKDM4ECYP1A2CYP2C19CYP2C9
SCHEMBL19979962 0.74 CYP1A2 (0.46) POLBKDM4ECYP1A2CYP2C19CYP2C9
SCHEMBL16719847 0.74 KMT2A (0.47) POLBKDM4ECYP1A2CYP2C19CYP2C9
SCHEMBL28396855 0.73 CYP1A2 (0.57) POLBKDM4ECYP1A2CYP2C19CYP2C9
SCHEMBL16719335 0.73 MYC (0.58) POLBKDM4ECYP1A2CYP2C19CYP2C9
SCHEMBL28608913 0.71 POLB (0.41) POLBKDM4EKMT2AALDH1A1TSHR
SCHEMBL16720403 0.71 OGT (0.45) KDM4ECYP1A2CYP2C19CYP2C9KMT2A
SCHEMBL1808749 0.71 ALDH1A1 (0.42) POLBKDM4ECYP1A2CYP2C19CYP2C9
SCHEMBL5869031 0.69 TP53 (0.64) POLBKDM4ECYP1A2CYP2C19CYP2C9
SCHEMBL3435440 0.69 OPRK1 (0.52) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111196804-A TGF- β R1 inhibitor and application thereof 南京圣和药业股份有限公司 2020-05-26 CN disclosed