SCHEMBL28643238

SCHEMBL28643238

COc1cccc(CN2CCCc3ccccc32)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.55
TSHR P16473 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
ALDH1A1 P00352 4/20 0.51
MAPK1 P28482 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
TMEM97 Q5BJF2 1/20 0.49
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
PTGER4 P35408 1/20 0.48
PTGER2 P43116 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.48
SIRT1 Q96EB6 1/20 0.48
HDAC1 Q13547 3/20 0.48
HDAC6 Q9UBN7 3/20 0.48
HDAC3 O15379 1/20 0.48
HDAC2 Q92769 1/20 0.48
ROCK2 O75116 1/20 0.48
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29483473 1.00 SIGMAR1 (0.55) SIGMAR1TSHRSMN1; SMN2ALDH1A1MAPK1
SCHEMBL5661589 0.92 SIGMAR1 (0.57) SIGMAR1TSHRALDH1A1TMEM97KDM4E
SCHEMBL29572755 0.92 SIGMAR1 (0.57) SIGMAR1TSHRALDH1A1TMEM97KDM4E
SCHEMBL29483476 0.85 ALDH1A1 (0.60) SIGMAR1TSHRSMN1; SMN2ALDH1A1MAPK1
SCHEMBL28743846 0.85 ALDH1A1 (0.60) SIGMAR1TSHRSMN1; SMN2ALDH1A1MAPK1
SCHEMBL29483475 0.82 BRD4 (0.55) TSHRSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL28642771 0.82 BRD4 (0.55) TSHRSMN1; SMN2ALDH1A1KDM4EMEN1
SCHEMBL1461825 0.80 HDAC1 (0.63) TSHRALDH1A1MAPK1L3MBTL1KDM4E
SCHEMBL29483474 0.80 HDAC1 (0.63) TSHRALDH1A1MAPK1L3MBTL1KDM4E
SCHEMBL16693159 0.80 KDM4E (0.59) TSHRSMN1; SMN2ALDH1A1MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112812060-B Arylation method of tetrahydroquinoline 绍兴文理学院 2022-04-29 CN disclosed
CN-112812060-A Arylation method of tetrahydroquinoline 绍兴文理学院 2021-05-18 CN disclosed