SCHEMBL28643265

SCHEMBL28643265

NC(=O)OCC1CCN(c2ccc(F)cc2C=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
FFAR4 Q5NUL3 2/20 0.38
CHRM3 P20309 9/20 0.38
RPS6KB1 P23443 2/20 0.36
MGLL Q99685 1/20 0.36
CHRM4 P08173 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28643274 0.93 RPS6KB1 (0.41) CHRM3RPS6KB1
SCHEMBL2557591 0.85 FFAR4 (0.41) FFAR4RPS6KB1CHRM4
SCHEMBL28659709 0.82 CHRM3 (0.34) CHRM3
SCHEMBL22781025 0.82 BPTF (0.48) FFAR4CHRM4
SCHEMBL28647168 0.81 MC4R (0.42) HDAC3HDAC1HDAC2FFAR4CHRM3
SCHEMBL28919339 0.80 CHRM4 (0.52) RPS6KB1CHRM4MAPT
SCHEMBL2560980 0.79 ALDH1A1 (0.49) MAPT
SCHEMBL28642501 0.75 CHRM3 (0.40) CHRM3RPS6KB1
SCHEMBL28653059 0.75 CHRM3 (0.40) CHRM3RPS6KB1
SCHEMBL28464943 0.74 ALDH1A1 (0.56) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113527298-A Macrocyclic lactam derivative, preparation method and application thereof 浙江海正药业股份有限公司 2021-10-22 CN disclosed